Publications

Papers in Refereed Journals

12. Arpin, Patrice; Hill, Bryan; Larouche-Gauthier, Robin; Spino, Claude “Prins cyclization of α-bromoethers under basic conditions” Canadian Journal of Chemistry, 2013, 91, 1193-1201.

http://www.nrcresearchpress.com/doi/pdf/10.1139/cjc-2013-0337

11. Hill, Bryan; Jordan, Robert; Qu, Yan;, Assoud, Abdeljalil; Rodrigo, Russell “A common synthetic route to homochiral tetracycles related to pillaromycinone and premithramycinone” Canadian Journal of Chemistry, 2011, 89, 1457-1468.

http://web.ebscohost.com/ehost/pdfviewer/pdfviewer?sid=1780206a-235b-49fd-997b-d655735e2985%40sessionmgr111&vid=2&hid=103

10. Ahmed, Ali M.; Hill, Bryan; Taylor, Scott D. “Trichloroethyl Group As a Protecting Group for Sulfonates and Its Application to the Synthesis of a Disulfonate Analog of the Tyrosine Sulfated PSGL-1 Peptide.” Journal of Organic Chemistry, 2009, 74, 3583-3586.

http://pubs.acs.org/doi/abs/10.1021/jo900122c

9. Hussain, M.; Ahmed, V.; Hill, B.; Taylor, S.D. “A re-examination of the difluoromethylenesulfonic acid group as a phosphotyrosine mimic for PTP1B inhibition” Bioorganic & Medicinal Chemistry, 2008, 16, 6764-6777.

http://www.sciencedirect.com/science/article/pii/S096808960800504X

8. Hill, B.; Ahmed, V.; Bates, D.; Taylor, S.D. “Enantioselective Synthesis of Protected L-4-[Sulfonamido(difluoromethyl)] phenylalanine and L-4-[Sulfonamido(methyl)]phenylalanine and an Examination of Hexa- and Tripeptide Platforms for Evaluating pTyr Mimics for PTP1B Inhibition.” Journal of Organic Chemistry, 2006, 71, 8190-8197

http://pubs.acs.org/doi/abs/10.1021/jo061496r

7. Hill, B.; Rodrigo, R. “Cyclohexenones as Michael Acceptors in the Staunton-Weinreb Annulation: A Simple Stannane Modification for the Synthesis of Polycyclic Systems” Organic Letters, 2005, 7(23), 5223-5225

http://pubs.acs.org/doi/abs/10.1021/ol052058u

6. Cecchi, A.; Taylor, S.D.; Liu, Y.; Hill, B.; Vullo, D.; Scozzafava, A.; Supuran, C.T. “Carbonic anhydrase inhibitors: Inhibition of human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides.” Bioorganic & Medicinal Chemistry Letters, 2005, 15, 5192-5196.

http://www.sciencedirect.com/science/article/pii/S0960894X05010966

5. Liu, Y.; Ahmed, V.; Hill, B.; Taylor, S.D. “Synthesis of a non-hydrolyzable estrone sulfate analogue bearing the difluoromethanesulfonamide group and its evaluation as a steroid sulfatase inhibitor.”  Organic & Biomolecular Chemistry, 2005, 3, 3329-3335.

http://pubs.rsc.org/en/content/articlepdf/2005/OB/B508852F

4. Hill, B.; Liu, Y.; Taylor, S.D. “Synthesis of a-Fluorosulfonamides by Electrophilic Fluorination.” Organic Letters, 2004, 6(23), 4285-4288.

http://pubs.acs.org/doi/abs/10.1021/ol048249z

3. Spino, C.; Hill, B.; Dubé, P.; Gingras, S. “A diene-transmissive approach to the quassinoid skeleton” Canadian Journal of Chemistry, 2003, 81, 81-108.

http://www.nrcresearchpress.com/doi/pdf/10.1139/v02-196

2. Hill, B.; De Vleeschauwer, M.; Houde, K.; Belley, M. “Aromatic Ring Opening of Fused Thiophenes via Organolithium Addition to Sulfur” SYNLETT 1998, 407-410.

1. Belley, M.L.; Hill, B.; Mitenko, H.; Scheigetz, J.; Zamboni, R. “Asymmetric Dihydroxylation of Dienes: Synthesis of Tetrols” SYNLETT 1996, 92-94.

Review Papers

1. Taylor, S.D.; Hill, B. “Recent advances in protein tyrosine phosphatase 1B inhibitors.” Expert opinion on investigational drugs. 2004, 13(3), 199-214.

http://informahealthcare.com/doi/abs/10.1517/13543784.13.3.199